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Found 3 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase kinase 3' and Ligand = 'BDBM50548192'
TargetMitogen-activated protein kinase kinase kinase kinase 3(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50548192(CHEMBL4749141)
Affinity DataIC50:  3nMAssay Description:Inhibition of GLK (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50548192(CHEMBL4749141)
Affinity DataIC50:  278nMAssay Description:Inhibition of GLK (unknown origin) transfected in human 293T cells co-transfected with GFP-fused PKCtheta assessed as reduction in PKCtheta phosphory...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50548192(CHEMBL4749141)
Affinity DataIC50:  434nMAssay Description:Inhibition of GLK in human T cells assessed as reduction in PKCtheta phosphorylation by Western blot analysisMore data for this Ligand-Target Pair