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Found 6 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50000655'
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655((4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  52nMAssay Description:Binding affinity against mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655((4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  52nMAssay Description:Binding affinity against mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655((4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655((4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  107nMAssay Description:Binding affinity against opioid receptor mu in guinea pig brain homogenates, using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655((4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  107nMAssay Description:Compound was tested for the inhibition of [3H]- [D-Ala2, N-MePhe4, Gly5-ol]-enkephalin (DAMGO) binding to Opioid receptor mu 1 in guinea pig brain ho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655((4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataIC50:  460nMAssay Description:Inhibitory concentration of compound against mu opioid receptor in guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed