TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 4.96E+3nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 7.81E+3nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 1.52E+4nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 156nMAssay Description:Tested for inhibition of amplification of electrically induced twitch in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair