TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing mu opioid receptorMore data for this Ligand-Target Pair