TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 522nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair