Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50045776'
TargetMu-type opioid receptor(Homo sapiens (Human))
St. John'S University

Curated by ChEMBL
LigandPNGBDBM50045776(CHEMBL982 | JF-1 | NALMEFENE | Nalmetrene | ORF-11...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]DAMGO from human mu-opioid receptor expressed in CHO cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045776(CHEMBL982 | JF-1 | NALMEFENE | Nalmetrene | ORF-11...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]-Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
St. John'S University

Curated by ChEMBL
LigandPNGBDBM50045776(CHEMBL982 | JF-1 | NALMEFENE | Nalmetrene | ORF-11...)
Affinity DataKi:  0.440nMAssay Description:Activity at human cloned mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
St. John'S University

Curated by ChEMBL
LigandPNGBDBM50045776(CHEMBL982 | JF-1 | NALMEFENE | Nalmetrene | ORF-11...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in HEK293 cells by visible spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed