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Found 4 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50071865'
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50071865((S)-2-Amino-N-(6-benzyl-1,2,3,4-tetrahydro-quinoli...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity against mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50071865((S)-2-Amino-N-(6-benzyl-1,2,3,4-tetrahydro-quinoli...)
Affinity DataKi:  2.62nMAssay Description:Binding affinity against Opioid receptor kappa 1 in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50071865((S)-2-Amino-N-(6-benzyl-1,2,3,4-tetrahydro-quinoli...)
Affinity DataEC50:  0.180nMAssay Description:Binding affinity against Opioid receptor delta 1 in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50071865((S)-2-Amino-N-(6-benzyl-1,2,3,4-tetrahydro-quinoli...)
Affinity DataEC50:  0.180nMAssay Description:Compound was tested for its ability to stimulate [35S]GTP-gamma-S, binding to membranes from C6 glioma cells stably expressing rat mu opioid receptor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed