TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences
Curated by ChEMBL
Mossakowski Medical Research Centre Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 0.740nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:In vitro binding affinity towards mu opioid receptors was determined using [3H]-[p-Cl-Phe]- 4] DPDPE or [3H]-Deltorphin IIMore data for this Ligand-Target Pair