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Found 2 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50081529'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50:  0.740nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50:  0.880nMAssay Description:In vitro binding affinity towards mu opioid receptors was determined using [3H]-[p-Cl-Phe]- 4] DPDPE or [3H]-Deltorphin IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed