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Found 3 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50101612'
TargetMu-type opioid receptor(GUINEA PIG)
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50101612(2-Amino-1-(3-benzyloxymethyl-3,4-dihydro-1H-isoqui...)
Affinity DataKi:  6.40nMAssay Description:Inhibition of guinea pig ileum Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50101612(2-Amino-1-(3-benzyloxymethyl-3,4-dihydro-1H-isoqui...)
Affinity DataIC50:  13nMAssay Description:Agonist potency using GTP-gamma [35S]- binding assay for mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50101612(2-Amino-1-(3-benzyloxymethyl-3,4-dihydro-1H-isoqui...)
Affinity DataEC50:  525nMAssay Description:Negative logarithm of the molar concentration for agonist activity at mu receptor was determined in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed