Affinity DataKi: 0.650nMAssay Description:Displacement of [3H]diprenorphine from rat mu opioid receptor transfected in C6 cells by liquid scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10nMAssay Description:Agonist activity at rat mu opioid receptor transfected in C6 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair