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Found 3 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50203825'
TargetMu-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50203825(CHEMBL375070 | Tyr-Pro-Phe-D-2-Nal-NH2)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-diprenorphine from human MOR expressed in CHO cell membranes after 80 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Medical University Of Lodz

Curated by ChEMBL
LigandPNGBDBM50203825(CHEMBL375070 | Tyr-Pro-Phe-D-2-Nal-NH2)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50203825(CHEMBL375070 | Tyr-Pro-Phe-D-2-Nal-NH2)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human MOR expressed in CHO cell membranes assessed as inhibition of CYM51010-induced [35S]-GTPgammaS binding preincubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed