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Found 2 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50297303'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50297303((S)-5-(1H-benzo[d]imidazol-2-yloxy)-4-((S)-2-((S)-...)
Affinity DataKi:  1.45nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50297303((S)-5-(1H-benzo[d]imidazol-2-yloxy)-4-((S)-2-((S)-...)
Affinity DataIC50:  494nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig longitudinal muscle myenteric plexus assessed as inhibition of electrically evoked contr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed