TargetMu-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.75nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair