Affinity DataKi: 0.600nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Activity was evaluated in human mu opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair