TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as induction of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair