TargetMu-type opioid receptor(Rattus norvegicus (rat))
Harbin Institute Of Technology
Curated by ChEMBL
Harbin Institute Of Technology
Curated by ChEMBL
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at mu-opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incub...More data for this Ligand-Target Pair