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Found 1 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50324363'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universita Degli Studi Di Torino

Curated by ChEMBL
LigandPNGBDBM50324363(4-Octyloxy-3-phenylsulfonylfuroxan | CHEMBL1215645)
Affinity DataEC50:  8.70E+3nMAssay Description:Inhibition of MRP1 expressed in MDCK cells assessed as calcein AM accumulation by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed