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Found 1 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50324378'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universita Degli Studi Di Torino

Curated by ChEMBL
LigandPNGBDBM50324378(3,4-diphenyl-1,2,5-oxadiazole 2-oxide | CHEMBL1212...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of MRP1 expressed in MDCK cells assessed as calcein AM accumulation by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed