Found 3 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50409816'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Laboratoire De Pharmacologie-Toxicologie Inra
Curated by ChEMBL
Laboratoire De Pharmacologie-Toxicologie Inra
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:TP_TRANSPORTER: inhibition of ATPase activity in Sf9 cells (membrane vesicles)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Laboratoire De Pharmacologie-Toxicologie Inra
Curated by ChEMBL
Laboratoire De Pharmacologie-Toxicologie Inra
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of Calcein-AM transport in HL60-MRP1 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Laboratoire De Pharmacologie-Toxicologie Inra
Curated by ChEMBL
Laboratoire De Pharmacologie-Toxicologie Inra
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of ATPase activity in Sf9 cells (membrane vesicles)More data for this Ligand-Target Pair