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Found 6 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50485609'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  0.765nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  6.32nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  110nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  162nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  1.63E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/MRP cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  3.05E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed