Found 6 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50485612'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 0.960nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 9.36nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 182nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 2.76E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/MRP cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 7.77E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair