Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1/M2/M3/M4/M5' and Ligand = 'BDBM50004726'
Affinity DataKi: 1.10nMAssay Description:Binding affinity to muscarinic acetylcholine receptor was determined in presence of [3H]OXO-M radioligand (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to muscarinic acetylcholine receptor was determined in presence of [3H]QNB radioligand (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
University Of Uppsala
Curated by ChEMBL
University Of Uppsala
Curated by ChEMBL
Affinity DataKd: 91nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair