Found 13 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1/M2/M3/M4/M5' and Ligand = 'BDBM50004734'
Affinity DataKi: 0.860nMAssay Description:Binding affinity to muscarinic acetylcholine receptor was determined in presence of [3H]OXO-M radioligand (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]CD as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to muscarinic acetylcholine receptor was determined in presence of [3H]QNB radioligand (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Dissociation constant for complex with muscarinic acetylcholine receptor M3 of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Compound was tested for the concentration that inhibited the specific binding of (-)-[3H]-NMS to muscarinic receptor in the rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding activity to muscarinic acetylcholine receptor in rat heart, assayed using [3H]-QNB as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding activity against Muscarinic acetylcholine receptor in rat cortex, using [3H]QNB as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide by filter plate assayMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity was determined using [3H]-NMS for Muscarinic acetylcholine receptor in SK-N-SH neuroblastoma cellsMore data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair