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Found 6 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1/M2/M3/M4/M5' and Ligand = 'BDBM50228577'
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKi:  170nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKi:  430nMAssay Description:Binding activity against Muscarinic acetylcholine receptor in rat cortex, using [3H]QNB as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKi:  450nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]CD as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKi:  610nMAssay Description:Binding activity to muscarinic acetylcholine receptor in rat heart, assayed using [3H]-QNB as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKi:  1.63E+3nMAssay Description:Binding activity to muscarinic acetylcholine receptor in rat heart, assayed using [3H]QNB as a radioligand in the presence of Gpp(NH)p.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKd:  1.16E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed