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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50038224'
TargetMuscarinic acetylcholine receptor M1(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50038224(5-(2-Ethyl-2H-[1,2,3]triazol-4-yl)-1-methyl-1,2,3,...)
Affinity DataKi:  24nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50038224(5-(2-Ethyl-2H-[1,2,3]triazol-4-yl)-1-methyl-1,2,3,...)
Affinity DataEC50: >1.20E+3nMAssay Description:M1 agonist activity estimated by rat superior cervical ganglion depolarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed