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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50061556'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50061556(11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]d...)
Affinity DataIC50:  37nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50061556(11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]d...)
Affinity DataIC50:  37nMAssay Description:Inhibitory binding of [3H]-pirenzepine to human Muscarinic acetylcholine receptor M1 in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed