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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50283129'
LigandPNGBDBM50283129(5-(4-Hex-3-ynyloxy-[1,2,5]thiadiazol-3-yl)-1,2-dim...)
Affinity DataIC50:  5nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 by the displacement of [3H]-pirenzepine in rat cerebral cortical membranesMore data for this Ligand-Target Pair
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LigandPNGBDBM50283129(5-(4-Hex-3-ynyloxy-[1,2,5]thiadiazol-3-yl)-1,2-dim...)
Affinity DataIC50:  6nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 by the displacement of [3H]-pirenzepine in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article