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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50121489'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121489((2-Amino-3-methyl-phenyl)-(4-{1-[4-(propane-2-sulf...)
Affinity DataKi:  0.890nMAssay Description:Binding affinity against cloned human muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121489((2-Amino-3-methyl-phenyl)-(4-{1-[4-(propane-2-sulf...)
Affinity DataKi:  6.60nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121489((2-Amino-3-methyl-phenyl)-(4-{1-[4-(propane-2-sulf...)
Affinity DataKi:  12nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121489((2-Amino-3-methyl-phenyl)-(4-{1-[4-(propane-2-sulf...)
Affinity DataKi:  12nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed