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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50246627'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246627(CHEMBL4065555)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M2 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50246627(CHEMBL4065555)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human recombinant muscarinic M2 receptor co-expressed with Galphaqi5-HA in African green monkey COS7 cells assessed as IP accumul...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed