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Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50417445'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Advanced Industrial Science And Technology (Aist)

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cell membranes incubated for 2 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Advanced Industrial Science And Technology (Aist)

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)
Affinity DataIC50:  0.158nMAssay Description:Displacement of [3H]NMS from recombinant human M2 receptor expressed in CHO-K1 cells after 16 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Advanced Industrial Science And Technology (Aist)

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)
Affinity DataIC50:  0.501nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed