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Found 10 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Ligand = 'BDBM50018056'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  820nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  838nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  1.26E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute of Mental Health

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  2.09E+3nMAssay Description:Binding affinity to human M3 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  4.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of rat submandibular muscarinic (M3) receptor isolated from tissue homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of rat submandibular muscarinic (M3) receptor isolated from tissue homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for glandular muscarinic acetylcholine receptor M3 in rat assayed using 0.3 nM [3H]N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for glandular muscarinic acetylcholine receptor M3 in rat assayed using 0.3 nM [3H]N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for glandular muscarinic acetylcholine receptor M3 in rat assayed using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed