Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50107696'
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  0.776nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity against M4 muscarinic receptor expressed in RBL-2H3 Mast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed