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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM502765'
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM502765((2S,6R)-4-(4-amino-5-cyanopyrimidin-2-yl)-N-[2-(1-...)
Affinity DataKi: >100nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM502765((2S,6R)-4-(4-amino-5-cyanopyrimidin-2-yl)-N-[2-(1-...)
Affinity DataKi: >100nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent