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Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM81901'
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  537nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]-NMS from human muscarinic M5 receptor expressed in stable CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  537nMMore data for this Ligand-Target Pair
In DepthDetails PubMed