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Found 4 Enz. Inhib. hit(s) with Target = 'Myosin light chain kinase family member 4' and Ligand = 'BDBM2579'
TargetMyosin light chain kinase family member 4(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  52.9nMAssay Description:Inhibition of human MYLK4 using KKRPQRRYSNVF as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase family member 4(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  54.5nMAssay Description:Inhibition of human MYLK4 using KKRPQRRYSNVF as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase family member 4(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  470nMAssay Description:Binding constant for MYLK4 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase family member 4(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  470nMAssay Description:Binding constant for SgK085 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed