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Found 4 Enz. Inhib. hit(s) with Target = 'N-alpha-acetyltransferase 40' and Ligand = 'BDBM50581153'
TargetN-alpha-acetyltransferase 40(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50581153(CHEMBL5081275)
Affinity DataKi:  0.610nMAssay Description:Competitive inhibition of human NatD using various concentration of human H4 peptide and fixed [14C]acetyl-CoA as substrate measured after 13 mins ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-alpha-acetyltransferase 40(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50581153(CHEMBL5081275)
Affinity DataKi:  1nMAssay Description:Inhibition of human NatD using H4-8 peptide substrate at Km value and AcCoA by Morrison's quadratic equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-alpha-acetyltransferase 40(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50581153(CHEMBL5081275)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of human NatD using H4-8 peptide substrate at 4 times Km value and AcCoA measured after 30 min incubation by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-alpha-acetyltransferase 40(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50581153(CHEMBL5081275)
Affinity DataIC50:  40nMAssay Description:Inhibition of human NatD using H4-8 peptide substrate at Km value and AcCoA measured after 30 min incubation by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed