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Found 2 Enz. Inhib. hit(s) with Target = 'N-arachidonyl glycine receptor' and Ligand = 'BDBM50221691'
TargetN-arachidonyl glycine receptor(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataIC50:  944nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment by measuring 2-(3-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-arachidonyl glycine receptor(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataEC50:  562nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed