Found 1 Enz. Inhib. hit(s) with Target = 'N-lysine methyltransferase KMT5A' and Ligand = 'BDBM50051129'
TargetN-lysine methyltransferase KMT5A(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
Curated by ChEMBL
University Of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of SETD8 (unknown origin) catalytic domain expressed in Escherichia coli using biotinylated H4 (1-24) peptide substrate after 1 hr by scin...More data for this Ligand-Target Pair