Found 2 Enz. Inhib. hit(s) with Target = 'N-lysine methyltransferase KMT5A' and Ligand = 'BDBM50201571'
Affinity DataKi: 50nMAssay Description:Competitive inhibition of human SETD8 (186 to 352 residues) using biotin-labeled H4K20 (1 to 24 residues) as substrate after 1 hr in presence of 3H-S...More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of human SETD8 (186 to 352 residues) using biotin-labeled H4K20 (1 to 24 residues) as substrate after 1 hr in presence of 3H-SAM by scinti...More data for this Ligand-Target Pair