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Found 2 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacetylase sirtuin-1' and Ligand = 'BDBM50392074'
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50392074(CHEMBL2152577)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of sirtuin 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50392074(CHEMBL2152577)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant SIRT1 using Fluor de Lys-SIRT as substrate incubated for 60 mins prior to substrate addition measured after 60 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed