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Found 2 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacetylase sirtuin-2' and Ligand = 'BDBM50228363'
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sirtris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50228363(CHEMBL257991 | N-(2-(3-(piperazin-1-ylmethyl)imida...)
Affinity DataEC50:  3.70E+4nMAssay Description:Activation of SIRT2 by mass spectrometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sirtris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50228363(CHEMBL257991 | N-(2-(3-(piperazin-1-ylmethyl)imida...)
Affinity DataEC50:  160nMAssay Description:Activation of human SirT2 protein fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed