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Found 3 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacylase sirtuin-5, mitochondrial' and Ligand = 'BDBM50576715'
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
The University Of Hong Kong

Curated by ChEMBL
LigandPNGBDBM50576715(CHEMBL4870282)
Affinity DataKi:  1.22E+5nMAssay Description:Inhibition of human recombinant SIRT5 assessed as inhibition of substrate desuccinylation using Fluor de Lys-Succinyl green peptide as substrate in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
The University Of Hong Kong

Curated by ChEMBL
LigandPNGBDBM50576715(CHEMBL4870282)
Affinity DataIC50:  1.83E+5nMAssay Description:Inhibition of human recombinant SIRT5 assessed as inhibition of substrate desuccinylation using Fluor de Lys-Succinyl green peptide as substrate in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
The University Of Hong Kong

Curated by ChEMBL
LigandPNGBDBM50576715(CHEMBL4870282)
Affinity DataKd:  2.47E+3nMAssay Description:Binding affinity to chip-immobilized recombinant human SIRT5 measured after 300 secs by surface plasmon resonance methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed