Affinity DataKi: 250nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in CHO cells assessed as inhibition of NKB-induced increase of intracellular calcium ...More data for this Ligand-Target Pair