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Found 2 Enz. Inhib. hit(s) with Target = 'Neuromedin-U receptor 2' and Ligand = 'BDBM50262112'
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50262112(CHEMBL4092080)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Mus musculus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50262112(CHEMBL4092080)
Affinity DataEC50:  0.75nMAssay Description:Agonist activity at mouse NMUR2 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed