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Found 1 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor; alpha9/alpha10' and Ligand = 'BDBM50339938'
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50339938(1,1',1'',1'''-(5,5',5'',5'''-(benzene-1,2,4,5-tetr...)
Affinity DataIC50:  5.40nMAssay Description:Antagonist activity at alpha9/alpha10 nAChR expressed in Xenopus oocyte assessed as inhibition of ACh-gated current by voltage clamp electrophysiolog...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed