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Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-3/beta-4' and Ligand = 'BDBM50139124'
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50139124(CHEMBL3759208)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-epibatidine from human alpha3beta4 nACh receptor expressed in HEK293 cells preincubated for 5 mins followed by radioligand addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50139124(CHEMBL3759208)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human alpha3beta4 nACh receptor expressed in rat GH4C1 cells assessed as increase in current amplitudes after 2 to 3 days by patc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed