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Found 1 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/beta-2' and Ligand = 'BDBM50382408'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382408(CHEMBL2022554)
Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed