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Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/beta-2' and Ligand = 'BDBM80642'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM80642(CHEMBL191491 | MG 624 | MLS002172460 | SMR00125409...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]-epibatidine from human alpha4beta2 nAChR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM80642(CHEMBL191491 | MG 624 | MLS002172460 | SMR00125409...)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of (+/-)-[3H]-epibatidine from human alpha4beta2 nAChR expressed in HEK293 cell membranes after 30 mins by beta counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed