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Found 1 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50078044'
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50078044(3-(6-Chloro-pyridin-3-ylmethyl)-3H-thiazol-(2E)-yl...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed