Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50279209'
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
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Curated by ChEMBL
LigandPNGBDBM50279209(CHEMBL498277 | N-[2-(Pyridin-2-yl)ethyl]cytisine)
Affinity DataKi:  941nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed